{"id":8911,"date":"2025-03-17T16:42:18","date_gmt":"2025-03-17T13:42:18","guid":{"rendered":"https:\/\/www.ortaakarsu.net\/?post_type=avada_portfolio&#038;p=8911"},"modified":"2025-04-26T19:35:10","modified_gmt":"2025-04-26T16:35:10","slug":"bir-bakteriyel-alarmon-enzimi-pppapp-sentetaz-pdb-8vx3","status":"publish","type":"avada_portfolio","link":"https:\/\/www.ortaakarsu.net\/?avada_portfolio=bir-bakteriyel-alarmon-enzimi-pppapp-sentetaz-pdb-8vx3","title":{"rendered":"Bir Bakteriyel Alarmon Enzimi &#8211; (p)ppApp Sentetaz (PDB 8VX3)"},"content":{"rendered":"<p><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-1 fusion-flex-container has-pattern-background has-mask-background hundred-percent-fullwidth non-hundred-percent-height-scrolling\" style=\"--awb-border-radius-top-left:0px;--awb-border-radius-top-right:0px;--awb-border-radius-bottom-right:0px;--awb-border-radius-bottom-left:0px;--awb-padding-top:0px;--awb-padding-bottom:0px;--awb-margin-bottom:-280px;--awb-background-color:var(--awb-color3);--awb-flex-wrap:wrap;\" ><div class=\"fusion-builder-row fusion-row fusion-flex-align-items-stretch fusion-flex-justify-content-space-evenly fusion-flex-content-wrap\" style=\"width:104% !important;max-width:104% !important;margin-left: calc(-4% \/ 2 );margin-right: calc(-4% \/ 2 );\"><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-0 fusion_builder_column_1_1 1_1 fusion-flex-column fusion-animated\" style=\"--awb-overflow:hidden;--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-border-radius:4px 4px 4px 4px;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:10px;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-spacing-right-medium:1.92%;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\" data-animationType=\"fadeInDown\" data-animationDuration=\"0.8\" data-animationOffset=\"top-into-view\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-video fusion-youtube\" style=\"--awb-max-width:1286px;--awb-max-height:720px;--awb-align-self:center;--awb-width:100%;--awb-margin-top:30px;\"><div class=\"video-shortcode\"><div class=\"fluid-width-video-wrapper\" style=\"padding-top:55.99%;\" ><iframe title=\"YouTube video player 1\" src=\"https:\/\/www.youtube.com\/embed\/-KJ4nDaJLtE?wmode=transparent&autoplay=0\" width=\"1286\" height=\"720\" allowfullscreen allow=\"autoplay; clipboard-write; encrypted-media; gyroscope; picture-in-picture;\"><\/iframe><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-1 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:32px;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-spacing-right-medium:1.92%;--awb-margin-bottom-medium:10px;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-title title fusion-title-1 fusion-sep-none fusion-title-marquee fusion-animate-once fusion-title-size-two\" style=\"--awb-text-color:var(--awb-color7);--awb-margin-bottom:6px;--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;--awb-marquee-speed:15000ms;--awb-marquee-translate-x:-100%;--awb-font-size:22px;\"><h2 class=\"fusion-title-heading title-heading-left awb-marquee-left\" style=\"margin:0;letter-spacing:0px;font-size:1em;\"><span class=\"awb-marquee-content\">Bir Bakteriyel Alarmon Enzimi \u2013 (p)ppApp Sentetaz (PDB 8VX3)<\/span><span class=\"awb-marquee-content\">Bir Bakteriyel Alarmon Enzimi \u2013 (p)ppApp Sentetaz (PDB 8VX3)<\/span><\/h2><\/div><div class=\"fusion-builder-row fusion-builder-row-inner fusion-row fusion-flex-align-items-stretch fusion-flex-justify-content-space-evenly fusion-flex-content-wrap\" style=\"--awb-flex-grow:0;--awb-flex-grow-medium:0;--awb-flex-grow-small:0;--awb-flex-shrink:0;--awb-flex-shrink-medium:0;--awb-flex-shrink-small:0;width:104% !important;max-width:104% !important;margin-left: 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8px;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:0px;--awb-margin-bottom-large:0px;--awb-spacing-left-large:0px;--awb-width-medium:100%;--awb-spacing-right-medium:0px;--awb-spacing-left-medium:0px;--awb-width-small:100%;--awb-spacing-right-small:0px;--awb-spacing-left-small:0px;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-title title fusion-title-2 fusion-sep-none fusion-title-text fusion-title-size-two\" style=\"--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;\"><h2 class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\"><h2>(p)ppApp Sentetaz Nedir?<\/h2><\/h2><\/div><div class=\"fusion-text fusion-text-2\" style=\"--awb-text-font-family:&quot;Nunito&quot;;--awb-text-font-style:normal;--awb-text-font-weight:400;\"><p><span class=\"fusion-dropcap dropcap\">S<\/span>treptomyces albidoflavus&#8217;tan (p)ppApp sentetaz analizimizle bakteriyel sava\u015f\u0131n molek\u00fcler d\u00fcnyas\u0131na dal\u0131n! Bu enzim bakteriyel bir alarmon sentetazd\u0131r &#8211; bir h\u00fccrenin metabolizmas\u0131n\u0131 saniyeler i\u00e7inde durdurabilen ola\u011fand\u0131\u015f\u0131 n\u00fckleotid habercileri olu\u015fturur. Kristal yap\u0131s\u0131n\u0131 (PDB ID: 8VX3) inceleyerek, \u015feklinin ve aktif b\u00f6lgesinin h\u00fccrenin enerji para birimini (ATP) ele ge\u00e7irmesine ve onu toksik bir sinyale d\u00f6n\u00fc\u015ft\u00fcrmesine nas\u0131l izin verdi\u011fini ortaya koyuyoruz.<\/p>\n<p>Bu videoda enzimin i\u015flevsel rol\u00fcn\u00fc a\u00e7\u0131kl\u0131yoruz: Bir fabrikan\u0131n g\u00fc\u00e7 jenerat\u00f6r\u00fcn\u00fcn aniden t\u00fcm elektri\u011fi hi\u00e7bir makinenin kullanamayaca\u011f\u0131 bir forma d\u00f6n\u00fc\u015ft\u00fcrd\u00fc\u011f\u00fcn\u00fc hayal edin &#8211; (p)ppApp&#8217;\u0131n bir bakteri h\u00fccresinde yapt\u0131\u011f\u0131 \u015fey budur. Bu enzim (p)ppApp \u00fcreterek ATP&#8217;yi (h\u00fccrenin \u201cpili\u201d) t\u00fcketir ve hayati s\u00fcre\u00e7leri durdurarak h\u00fccre \u00fczerindeki \u201ckapatma d\u00fc\u011fmesini\u201d etkili bir \u015fekilde kapat\u0131r. Ayr\u0131ca, bir bakterinin rakibinin altyap\u0131s\u0131n\u0131 nas\u0131l sabote edebilece\u011fini g\u00f6stermek i\u00e7in bir \u015fehir kesintisine benzetme yap\u0131yoruz. Bu (p)ppApp sentetaz genellikle bakteriler aras\u0131 rekabette bir toksin olarak kullan\u0131l\u0131r, yani bakteriler bunu kom\u015fular\u0131na kar\u015f\u0131 bir silah olarak kullan\u0131r. Bu ak\u0131ll\u0131ca bir stratejinin par\u00e7as\u0131d\u0131r: enzim bir rakibe enjekte edilerek kurban\u0131n enerjisinin t\u00fckenmesine ve b\u00fcy\u00fcmesinin durmas\u0131na neden olur.<\/p>\n<\/div><div class=\"fusion-text fusion-text-3\" style=\"--awb-text-font-family:&quot;Nunito&quot;;--awb-text-font-style:normal;--awb-text-font-weight:400;\"><p>Daha sonra, enzimin ba\u011flanma b\u00f6lgelerini ve katalitik kal\u0131nt\u0131lar\u0131n\u0131 yak\u0131nla\u015ft\u0131r\u0131yoruz. 3D yap\u0131, iki n\u00fckleotid i\u00e7in m\u00fckemmel boyutta bir cep g\u00f6steriyor: biri pirofosfat verirken di\u011feri (bir ADP veya ATP) onu al\u0131yor. Aktif b\u00f6lgedeki kilit bir amino asit, al\u0131c\u0131 molek\u00fcl\u00fcn 3\u2032-OH grubunu aktive etmek i\u00e7in katalitik bir baz g\u00f6revi g\u00f6rerek ATP&#8217;den bir pirofosfat\u0131n transferini sa\u011flar. Bu s\u00fcreci, enzimin ATP&#8217;den pirofosfat\u0131 almak i\u00e7in substrat\u0131 haz\u0131rlad\u0131\u011f\u0131 bir yar\u0131\u015ftaki bayrak teslimine benzetiyoruz. \u00d6zel olarak tasarlanm\u0131\u015f aktif b\u00f6lgesi sayesinde enzim \u00f6zellikle adenozin bazl\u0131 molek\u00fclleri hedef alarak (p)ppGpp yerine (p)ppApp yapmas\u0131n\u0131 sa\u011flar.<\/p>\n<p>Ayr\u0131ca ilgili proteinlerle yap\u0131sal kar\u015f\u0131la\u015ft\u0131rmalar\u0131 da vurguluyoruz. (p)ppApp sentetaz 207 amino asitlik tek bir protein olmas\u0131na ra\u011fmen, aktif durumda bir homotetramer olu\u015fturur. Bu yap\u0131, t\u00fcm par\u00e7alar\u0131n uyum i\u00e7inde \u00e7al\u0131\u015fmas\u0131 gereken \u00e7ok motorlu bir sistemi an\u0131msat\u0131r. Birden fazla etki alan\u0131na sahip olan ve ikili roller \u00fcstlenen daha b\u00fcy\u00fck RelA\/SpoT proteinlerinin aksine, Streptomyces enzimi yaln\u0131zca senteze adanm\u0131\u015f bir uzmand\u0131r ve bu da onu son derece verimli k\u0131lar. H\u0131zl\u0131 bir \u015fekilde alarmon molek\u00fclleri \u00fcretme kabiliyeti onu mikrobiyal rekabette g\u00fc\u00e7l\u00fc bir ara\u00e7 haline getirmektedir.<\/p>\n<p>Son olarak, enzimin daha geni\u015f biyolojik \u00f6nemini tart\u0131\u015f\u0131yoruz. (p)ppApp sentetaz, bakterilerde yeni bir n\u00fckleotid ikinci haberci sistemini temsil etmektedir. Yap\u0131s\u0131n\u0131n ve i\u015flevinin anla\u015f\u0131lmas\u0131, yenilik\u00e7i antibiyotik stratejilerinin veya biyoteknolojik uygulamalar\u0131n \u00f6n\u00fcn\u00fc a\u00e7abilir. Bu b\u00fcy\u00fcleyici enzimin molek\u00fcler dinamiklerini canland\u0131r\u0131rken, ayr\u0131nt\u0131l\u0131 yap\u0131sal bilgileri mikrobiyal hayatta kalma ve rekabet i\u00e7in ger\u00e7ek d\u00fcnyadaki sonu\u00e7larla ili\u015fkilendirirken bize kat\u0131l\u0131n.<\/p>\n<\/div><div class=\"fusion-text fusion-text-4\" style=\"--awb-text-font-family:&quot;Nunito&quot;;--awb-text-font-style:normal;--awb-text-font-weight:400;\"><h4>Referanslar<\/h4>\n<ul>\n<li>Bartoli, J., Tempier, A. C., Guzzi, N. L., Piras, C. M., Cascales, E., &amp; Viala, J. P. (2023). Characterization of a (p) ppApp Synthetase Belonging to a New Family of Polymorphic Toxin Associated with Temperate Phages. Journal of Molecular Biology, 435(21), 168282. <a href=\"https:\/\/doi.org\/10.1016\/j.jmb.2023.168282\">https:\/\/doi.org\/10.1016\/j.jmb.2023.168282<\/a><\/li>\n<li>Ahmad, S., Wang, B., Walker, M. D., Tran, H. K. R., Stogios, P. J., Savchenko, A., &#8230; &amp; Whitney, J. C. (2019). An interbacterial toxin inhibits target cell growth by synthesizing (p) ppApp. Nature, 575(7784), 674-678. <a href=\"https:\/\/www.nature.com\/articles\/s41586-019-1735-9\">https:\/\/www.nature.com\/articles\/s41586-019-1735-9<\/a><\/li>\n<\/ul>\n<\/div><\/div><\/div><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-5 fusion_builder_column_1_1 1_1 fusion-flex-column fusion-animated\" style=\"--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:0px;--awb-margin-bottom-large:40px;--awb-spacing-left-large:0px;--awb-width-medium:100%;--awb-spacing-right-medium:0px;--awb-spacing-left-medium:0px;--awb-width-small:100%;--awb-spacing-right-small:0px;--awb-spacing-left-small:0px;\" data-animationType=\"fadeInDown\" data-animationDuration=\"0.6\" data-animationOffset=\"top-into-view\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-sharing-box fusion-sharing-box-1 has-taglines layout-floated layout-medium-floated layout-small-floated\" style=\"background-color:var(--awb-color2);--awb-layout:row;--awb-alignment-small:space-between;\" data-title=\"Aktif B\u00f6lgeye G\u00f6m\u00fcl\u00fc Bir Ligand\u0131n Zamana Ba\u011fl\u0131 Hareketi\" data-description=\"Edible Easter Slime  Recommended for you    MMolek\u00fcler dinamik (MD) sim\u00fclasyonlar\u0131, geleneksel deneysel y\u00f6ntemlere gizli kalan atomik d\u00fczeydeki olaylar\u0131 g\u00f6rselle\u015ftirme ve anlama kapasitemizde devrim yaratm\u0131\u015ft\u0131r. 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