{"id":9030,"date":"2025-03-19T02:06:11","date_gmt":"2025-03-18T23:06:11","guid":{"rendered":"https:\/\/www.ortaakarsu.net\/?post_type=avada_portfolio&#038;p=9030"},"modified":"2025-03-19T02:20:25","modified_gmt":"2025-03-18T23:20:25","slug":"3d-simulasyon-nst-628-raf-mek-kompleksindeki-ras-mapk-yolagini-hedefliyor-guclu-kanser-tedavisi","status":"publish","type":"avada_portfolio","link":"https:\/\/www.ortaakarsu.net\/?avada_portfolio=3d-simulasyon-nst-628-raf-mek-kompleksindeki-ras-mapk-yolagini-hedefliyor-guclu-kanser-tedavisi","title":{"rendered":"3D Sim\u00fclasyon: NST-628, RAF-MEK Kompleksindeki RAS-MAPK Yola\u011f\u0131n\u0131 Hedefliyor | G\u00fc\u00e7l\u00fc Kanser Tedavisi"},"content":{"rendered":"<p><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-1 fusion-flex-container has-pattern-background has-mask-background hundred-percent-fullwidth non-hundred-percent-height-scrolling\" style=\"--awb-border-radius-top-left:0px;--awb-border-radius-top-right:0px;--awb-border-radius-bottom-right:0px;--awb-border-radius-bottom-left:0px;--awb-padding-top:0px;--awb-padding-bottom:0px;--awb-margin-bottom:-280px;--awb-background-color:var(--awb-color3);--awb-flex-wrap:wrap;\" ><div class=\"fusion-builder-row fusion-row fusion-flex-align-items-stretch fusion-flex-justify-content-space-evenly fusion-flex-content-wrap\" style=\"width:104% !important;max-width:104% !important;margin-left: calc(-4% \/ 2 );margin-right: calc(-4% \/ 2 );\"><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-0 fusion_builder_column_1_1 1_1 fusion-flex-column fusion-animated\" style=\"--awb-overflow:hidden;--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-border-radius:4px 4px 4px 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allow=\"autoplay; clipboard-write; encrypted-media; gyroscope; picture-in-picture;\"><\/iframe><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-1 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:32px;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-spacing-right-medium:1.92%;--awb-margin-bottom-medium:10px;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-title title fusion-title-1 fusion-sep-none fusion-title-marquee fusion-animate-once fusion-title-size-two\" style=\"--awb-text-color:var(--awb-color7);--awb-margin-bottom:6px;--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;--awb-marquee-speed:15000ms;--awb-marquee-translate-x:-100%;--awb-font-size:22px;\"><h2 class=\"fusion-title-heading title-heading-left awb-marquee-left\" style=\"margin:0;letter-spacing:0px;font-size:1em;\"><span class=\"awb-marquee-content\">3D Sim\u00fclasyon: NST-628, RAF-MEK Kompleksindeki RAS-MAPK Yola\u011f\u0131n\u0131 Hedefliyor | G\u00fc\u00e7l\u00fc Kanser Tedavisi<\/span><span class=\"awb-marquee-content\">3D Sim\u00fclasyon: NST-628, RAF-MEK Kompleksindeki RAS-MAPK Yola\u011f\u0131n\u0131 Hedefliyor | G\u00fc\u00e7l\u00fc Kanser Tedavisi<\/span><\/h2><\/div><div class=\"fusion-builder-row fusion-builder-row-inner fusion-row fusion-flex-align-items-stretch fusion-flex-justify-content-space-evenly fusion-flex-content-wrap\" 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href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=bir-bromodomain-inhibitoru-ile-sitma-ilacini-kesfetmek-bir-molekuler-dinamik-simulasyonu\" aria-label=\"Bir Bromodomain \u0130nhibit\u00f6r\u00fc ile S\u0131tma \u0130lac\u0131n\u0131 Ke\u015ffetmek: Bir Molek\u00fcler Dinamik Sim\u00fclasyonu\"><\/a>\n\t<\/div>\n<\/div>\n<\/div>\n<h4 class=\"fusion-carousel-title\"><a href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=bir-bromodomain-inhibitoru-ile-sitma-ilacini-kesfetmek-bir-molekuler-dinamik-simulasyonu\" target=\"_self\">Bir Bromodomain \u0130nhibit\u00f6r\u00fc ile S\u0131tma \u0130lac\u0131n\u0131 Ke\u015ffetmek: Bir Molek\u00fcler Dinamik Sim\u00fclasyonu<\/a><\/h4><div class=\"fusion-carousel-meta\"><a href=\"https:\/\/www.ortaakarsu.net\/?portfolio_category=molekuler-dinamik-videolari\" rel=\"tag\">Molek\u00fcler Dinamik Videolar\u0131<\/a><\/div><\/div><\/div><div class=\"swiper-slide\"><div class=\"fusion-carousel-item-wrapper\"><span class=\"entry-title 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https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/glikozidaz_serit_fon-1-1200x675.png 1200w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/glikozidaz_serit_fon-1.png 1920w\" sizes=\"(min-width: 2200px) 100vw, (min-width: 856px) 278px, (min-width: 784px) 370px, (min-width: 712px) 555px, (min-width: 640px) 712px, \" \/><div class=\"fusion-rollover\">\n\t<div class=\"fusion-rollover-content\">\n\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t<a class=\"fusion-rollover-link\" href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=bir-bakteriyel-alarmon-enzimi-pppapp-sentetaz-pdb-8vx3\">Bir Bakteriyel Alarmon Enzimi &#8211; (p)ppApp Sentetaz (PDB 8VX3)<\/a>\n\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\n\t\t\t\t\t\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t<div class=\"fusion-rollover-sep\"><\/div>\n\t\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<a class=\"fusion-rollover-gallery\" href=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/glikozidaz_serit_fon-1.png\" data-options=\"\" data-id=\"8911\" 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href=\"https:\/\/www.ortaakarsu.net\/?portfolio_category=molekuler-dinamik-videolari\" rel=\"tag\">Molek\u00fcler Dinamik Videolar\u0131<\/a><\/div><\/div><\/div><div class=\"swiper-slide\"><div class=\"fusion-carousel-item-wrapper\"><span class=\"entry-title rich-snippet-hidden\">AMPK&#8217;n\u0131n \u00c7arp\u0131c\u0131 4K Molek\u00fcler Dinami\u011fi (PDB 3AQV) | Bilim Sanatla Bulu\u015fuyor<\/span><span class=\"vcard rich-snippet-hidden\"><span class=\"fn\"><a href=\"https:\/\/www.ortaakarsu.net\/?author=1\" rel=\"author\">ORTAAKARSU<\/a><\/span><\/span><span class=\"updated rich-snippet-hidden\">2025-03-18T15:33:45+03:00<\/span><div  class=\"fusion-image-wrapper\" aria-haspopup=\"true\">\n\t\t\t\t<img decoding=\"async\" width=\"1920\" height=\"1080\" src=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/tetramer_fon-1.png\" class=\"attachment-full size-full wp-post-image\" alt=\"\" srcset=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/tetramer_fon-1-200x113.png 200w, 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Bulu\u015fuyor<\/a>\n\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\n\t\t\t\t\t\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t<div class=\"fusion-rollover-sep\"><\/div>\n\t\t\t\t\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<a class=\"fusion-rollover-gallery\" href=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/tetramer_fon-1.png\" data-options=\"\" data-id=\"8903\" data-rel=\"iLightbox[gallery-rw-1]\" data-title=\"tetramer_fon (1)\" data-caption=\"\">\n\t\t\t\t\t\tGallery\t\t\t\t\t<\/a>\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\n\t\t\n\t\t\t\t\t\t\t\t\n\t\t\t\t\t\t\t\t\t\t<div class=\"fusion-rollover-categories\"><a href=\"https:\/\/www.ortaakarsu.net\/?portfolio_category=molekuler-dinamik-videolari\" rel=\"tag\">Molek\u00fcler Dinamik Videolar\u0131<\/a><\/div>\t\t\t\t\t\n\t\t\n\t\t\t\t\t\t<a class=\"fusion-link-wrapper\" href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=ampknin-carpici-4k-molekuler-dinamigi-pdb-3aqv-bilim-sanatla-bulusuyor\" aria-label=\"AMPK&#8217;n\u0131n \u00c7arp\u0131c\u0131 4K Molek\u00fcler Dinami\u011fi (PDB 3AQV) | Bilim Sanatla Bulu\u015fuyor\"><\/a>\n\t<\/div>\n<\/div>\n<\/div>\n<h4 class=\"fusion-carousel-title\"><a href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=ampknin-carpici-4k-molekuler-dinamigi-pdb-3aqv-bilim-sanatla-bulusuyor\" target=\"_self\">AMPK&#8217;n\u0131n \u00c7arp\u0131c\u0131 4K Molek\u00fcler Dinami\u011fi (PDB 3AQV) | Bilim Sanatla Bulu\u015fuyor<\/a><\/h4><div class=\"fusion-carousel-meta\"><a href=\"https:\/\/www.ortaakarsu.net\/?portfolio_category=molekuler-dinamik-videolari\" rel=\"tag\">Molek\u00fcler Dinamik Videolar\u0131<\/a><\/div><\/div><\/div><div class=\"swiper-slide\"><div class=\"fusion-carousel-item-wrapper\"><span class=\"entry-title rich-snippet-hidden\">Alfa-Glukozidaz&#8217;da Allosterik \u0130nhibisyon: 4K Hiper-Ger\u00e7ek\u00e7i Molek\u00fcler Dinamik Sim\u00fclasyonu<\/span><span class=\"vcard rich-snippet-hidden\"><span class=\"fn\"><a href=\"https:\/\/www.ortaakarsu.net\/?author=1\" rel=\"author\">ORTAAKARSU<\/a><\/span><\/span><span class=\"updated rich-snippet-hidden\">2025-03-18T15:38:34+03:00<\/span><div  class=\"fusion-image-wrapper\" aria-haspopup=\"true\">\n\t\t\t\t<img decoding=\"async\" width=\"1920\" height=\"1080\" src=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i.png\" class=\"attachment-full size-full wp-post-image\" alt=\"\" srcset=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i-200x113.png 200w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i-400x225.png 400w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i-600x338.png 600w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i-800x450.png 800w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/amilaz_substrat_alosterik_inhib12i-1200x675.png 1200w, 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href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=aktif-bolgeye-gomulu-bir-ligandin-zamana-bagli-hareketi\" aria-label=\"Aktif B\u00f6lgeye G\u00f6m\u00fcl\u00fc Bir Ligand\u0131n Zamana Ba\u011fl\u0131 Hareketi\"><\/a>\n\t<\/div>\n<\/div>\n<\/div>\n<h4 class=\"fusion-carousel-title\"><a href=\"https:\/\/www.ortaakarsu.net\/?avada_portfolio=aktif-bolgeye-gomulu-bir-ligandin-zamana-bagli-hareketi\" target=\"_self\">Aktif B\u00f6lgeye G\u00f6m\u00fcl\u00fc Bir Ligand\u0131n Zamana Ba\u011fl\u0131 Hareketi<\/a><\/h4><div class=\"fusion-carousel-meta\"><a href=\"https:\/\/www.ortaakarsu.net\/?portfolio_category=molekuler-dinamik-videolari\" rel=\"tag\">Molek\u00fcler Dinamik Videolar\u0131<\/a><\/div><\/div><\/div><\/div><div class=\"awb-swiper-button awb-swiper-button-prev\"><i class=\"awb-icon-angle-left\" aria-hidden=\"true\"><\/i><\/div><div class=\"awb-swiper-button awb-swiper-button-next\"><i class=\"awb-icon-angle-right\" aria-hidden=\"true\"><\/i><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-3 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:1.92%;--awb-margin-bottom-large:0%;--awb-spacing-left-large:1.92%;--awb-width-medium:100%;--awb-spacing-right-medium:1.92%;--awb-spacing-left-medium:1.92%;--awb-width-small:100%;--awb-spacing-right-small:1.92%;--awb-spacing-left-small:1.92%;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-separator fusion-full-width-sep\" style=\"align-self: center;margin-left: auto;margin-right: auto;margin-top:10%;margin-bottom:80px;width:100%;\"><div class=\"fusion-separator-border sep-shadow\" style=\"--awb-height:20px;--awb-amount:20px;background:radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-webkit-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-moz-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-o-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);\"><\/div><\/div><div class=\"fusion-section-separator section-separator big-half-circle fusion-section-separator-1\" style=\"--awb-spacer-height:99px;--awb-svg-margin-left:1.92%;--awb-svg-margin-right:1.92%;--awb-svg-margin-left-medium:1.92%;--awb-svg-margin-right-medium:1.92%;--awb-svg-margin-left-small:1.92%;--awb-svg-margin-right-small:1.92%;--awb-divider-height:99px;--awb-spacer-padding-top:inherit;--awb-sep-padding:0;--awb-svg-padding:0;\"><div class=\"fusion-section-separator-svg\"><svg class=\"fusion-big-half-circle-candy\" xmlns=\"http:\/\/www.w3.org\/2000\/svg\" version=\"1.1\" width=\"100%\" height=\"100\" viewBox=\"0 0 100 100\" preserveAspectRatio=\"none\" fill=\"rgba(249,249,251,1)\"><path d=\"M0 100 C40 0 60 0 100 100 Z\"><\/path><\/svg><\/div><div class=\"fusion-section-separator-spacer\"><div class=\"fusion-section-separator-spacer-height\"><\/div><\/div><\/div><\/div><\/div><\/div><\/div><div class=\"fusion-fullwidth fullwidth-box fusion-builder-row-2 fusion-flex-container nonhundred-percent-fullwidth non-hundred-percent-height-scrolling\" style=\"--awb-border-radius-top-left:0px;--awb-border-radius-top-right:0px;--awb-border-radius-bottom-right:0px;--awb-border-radius-bottom-left:0px;--awb-padding-top:0px;--awb-padding-bottom:0px;--awb-flex-wrap:wrap;\" ><div class=\"fusion-builder-row fusion-row fusion-flex-align-items-flex-start fusion-flex-content-wrap\" style=\"max-width:calc( 1200px + 0px );margin-left: calc(-0px \/ 2 );margin-right: calc(-0px \/ 2 );\"><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-4 fusion_builder_column_1_1 1_1 fusion-flex-column\" style=\"--awb-padding-top:8%;--awb-padding-right:10%;--awb-padding-bottom:5%;--awb-padding-left:10%;--awb-padding-right-medium:60px;--awb-padding-left-medium:60px;--awb-padding-right-small:40px;--awb-padding-left-small:40px;--awb-overflow:hidden;--awb-bg-color:var(--awb-color1);--awb-bg-color-hover:var(--awb-color1);--awb-bg-size:cover;--awb-box-shadow:0px 10px 63px 38px hsla(var(--awb-color7-h),var(--awb-color7-s),var(--awb-color7-l),calc( var(--awb-color7-a) - 93% ));;--awb-border-radius:8px 8px 8px 8px;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:0px;--awb-margin-bottom-large:0px;--awb-spacing-left-large:0px;--awb-width-medium:100%;--awb-spacing-right-medium:0px;--awb-spacing-left-medium:0px;--awb-width-small:100%;--awb-spacing-right-small:0px;--awb-spacing-left-small:0px;\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-text fusion-text-2 awb-text-cols fusion-text-columns-2\" style=\"--awb-columns:2;--awb-column-spacing:2em;--awb-column-min-width:100px;--awb-text-font-family:&quot;Nunito&quot;;--awb-text-font-style:normal;--awb-text-font-weight:400;\"><p><span class=\"fusion-dropcap dropcap\">B<\/span>RAF\/MEK kompleksinin kristal yap\u0131s\u0131na (PDB ID: 9AXY) dayanan bu geli\u015fmi\u015f, ger\u00e7ek\u00e7i 3D sim\u00fclasyon arac\u0131l\u0131\u011f\u0131yla yenilik\u00e7i molek\u00fcler yap\u0131\u015ft\u0131r\u0131c\u0131 NST-628&#8217;in karma\u015f\u0131k molek\u00fcler dinamiklerini ke\u015ffedin. NST-628, \u00e7ok say\u0131da solid t\u00fcm\u00f6r ve agresif kanserde \u00f6nemli bir etken olan RAS-MAPK sinyal yolunu g\u00fc\u00e7l\u00fc bir \u015fekilde hedeflemek ve bask\u0131lamak i\u00e7in tasarlanm\u0131\u015f \u00f6nc\u00fc bir pan-RAF-MEK inhibit\u00f6r\u00fcd\u00fcr.<\/p>\n<\/div><div class=\"fusion-title title fusion-title-2 fusion-sep-none fusion-title-text fusion-title-size-two\" style=\"--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;\"><h2 class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\"><h2>BRAF\/MEK Yola\u011f\u0131<\/h2><\/h2><\/div><div class=\"fusion-text fusion-text-3 awb-text-cols fusion-text-columns-2\" style=\"--awb-columns:2;--awb-column-spacing:2em;--awb-column-min-width:100px;\"><p>Derinlemesine yap\u0131sal analiz ve biyokimyasal \u00e7al\u0131\u015fmalar, NST-628&#8217;in RAF-MEK kompleksi i\u00e7indeki inaktif konformasyonlar\u0131 etkili bir \u015fekilde stabilize etti\u011fini do\u011frulamaktad\u0131r. Bu stabilizasyon, mevcut hedefe y\u00f6nelik kanser tedavilerinde s\u0131kl\u0131kla kar\u015f\u0131la\u015f\u0131lan diren\u00e7 mekanizmalar\u0131n\u0131n \u00fcstesinden gelerek derin ve s\u00fcrekli yol inhibisyonuna yol a\u00e7maktad\u0131r. \u00d6zellikle, NST-628 ola\u011fan\u00fcst\u00fc kan-beyin bariyeri ge\u00e7irgenli\u011fine sahiptir ve intrakraniyal t\u00fcm\u00f6rler ve merkezi sinir sistemi tutulumu olan kanserler i\u00e7in umut verici bir terap\u00f6tik potansiyel sunar.<\/p>\n<\/div><div class=\"fusion-title title fusion-title-3 fusion-sep-none fusion-title-text fusion-title-size-three\" style=\"--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;\"><h3 class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\"><h3>\u0130la\u00e7 Tasar\u0131m<\/h3><\/h3><\/div><div class=\"fusion-text fusion-text-4 awb-text-cols fusion-text-columns-2\" style=\"--awb-columns:2;--awb-column-spacing:2em;--awb-column-min-width:100px;\"><p>Titiz h\u00fccresel deneylerde ve \u00e7e\u015fitli hasta kaynakl\u0131 t\u00fcm\u00f6r ksenograft modellerinde NST-628, zorlu ortotopik intrakraniyal modeller de dahil olmak \u00fczere \u00e7e\u015fitli MAPK yola\u011f\u0131 mutasyonlar\u0131n\u0131 bar\u0131nd\u0131ran t\u00fcm\u00f6rlere kar\u015f\u0131 geni\u015f spektrumlu etkinlik g\u00f6stermi\u015ftir. Bile\u015fi\u011fin farmakokinetik profili, g\u00fc\u00e7l\u00fc beyin penetrasyonunu vurgulamakta ve onu onkolojide d\u00f6n\u00fc\u015ft\u00fcr\u00fcc\u00fc bir terap\u00f6tik aday olarak konumland\u0131rmaktad\u0131r.<\/p>\n<\/div><div class=\"fusion-separator fusion-full-width-sep\" style=\"align-self: center;margin-left: auto;margin-right: auto;margin-top:32px;width:100%;\"><div class=\"fusion-separator-border sep-shadow\" style=\"--awb-height:20px;--awb-amount:20px;background:radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-webkit-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-moz-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-o-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);\"><\/div><\/div><div class=\"fusion-image-element\" style=\"text-align:center;--awb-max-width:600px;--awb-caption-title-font-family:var(--h2_typography-font-family);--awb-caption-title-font-weight:var(--h2_typography-font-weight);--awb-caption-title-font-style:var(--h2_typography-font-style);--awb-caption-title-size:var(--h2_typography-font-size);--awb-caption-title-transform:var(--h2_typography-text-transform);--awb-caption-title-line-height:var(--h2_typography-line-height);--awb-caption-title-letter-spacing:var(--h2_typography-letter-spacing);\"><span class=\" fusion-imageframe imageframe-none imageframe-1 hover-type-magnify has-image-magnify fusion-animated\" style=\"border-radius:10px;\" data-animationType=\"fadeInDown\" data-animationDuration=\"0.4\" data-animationOffset=\"top-into-view\" data-magnify-duration=\"400\"><img decoding=\"async\" width=\"1024\" height=\"576\" title=\"molecule_zoom (1)\" src=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-1024x576.png\" alt class=\"img-responsive wp-image-8997\" srcset=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-200x112.png 200w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-400x225.png 400w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-600x337.png 600w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-800x450.png 800w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/molecule_zoom-1-1200x675.png 1200w\" sizes=\"(max-width: 640px) 100vw, 1200px\" \/><\/span><\/div><div class=\"fusion-separator fusion-full-width-sep\" style=\"align-self: center;margin-left: auto;margin-right: auto;margin-top:30px;width:100%;\"><div class=\"fusion-separator-border sep-shadow\" style=\"--awb-height:20px;--awb-amount:20px;background:radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-webkit-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-moz-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-o-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);\"><\/div><\/div><div class=\"fusion-title title fusion-title-4 fusion-sep-none fusion-title-text fusion-title-size-four\" style=\"--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;\"><h4 class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\">\u0130naktif Konformasyonun Stabilizasyonu<\/h4><\/div><div class=\"fusion-text fusion-text-5 awb-text-cols fusion-text-columns-2\" style=\"--awb-columns:2;--awb-column-spacing:2em;--awb-column-min-width:100px;\"><p>Derinlemesine yap\u0131sal analiz ve biyokimyasal \u00e7al\u0131\u015fmalar, NST-628&#8217;in RAF-MEK kompleksi i\u00e7indeki inaktif konformasyonlar\u0131 etkili bir \u015fekilde stabilize etti\u011fini do\u011frulamaktad\u0131r. Bu stabilizasyon, mevcut hedefe y\u00f6nelik kanser tedavilerinde s\u0131kl\u0131kla kar\u015f\u0131la\u015f\u0131lan diren\u00e7 mekanizmalar\u0131n\u0131n \u00fcstesinden gelerek derin ve s\u00fcrekli yol inhibisyonuna yol a\u00e7maktad\u0131r. \u00d6zellikle, NST-628 ola\u011fan\u00fcst\u00fc kan-beyin bariyeri ge\u00e7irgenli\u011fine sahiptir ve intrakraniyal t\u00fcm\u00f6rler ve merkezi sinir sistemi tutulumu olan kanserler i\u00e7in umut verici bir terap\u00f6tik potansiyel sunar.<\/p>\n<p><span style=\"color: var(--awb-text-color); font-family: var(--awb-text-font-family); font-size: var(--awb-font-size); font-style: var(--awb-text-font-style); font-weight: var(--awb-text-font-weight); letter-spacing: var(--awb-letter-spacing); text-align: var(--awb-content-alignment); text-transform: var(--awb-text-transform); background-color: var(--awb-bg-color-medium-hover);\">Titiz h\u00fccresel deneylerde ve \u00e7e\u015fitli hasta kaynakl\u0131 t\u00fcm\u00f6r ksenograft modellerinde NST-628, zorlu ortotopik intrakraniyal modeller de dahil olmak \u00fczere \u00e7e\u015fitli MAPK yola\u011f\u0131 mutasyonlar\u0131n\u0131 bar\u0131nd\u0131ran t\u00fcm\u00f6rlere kar\u015f\u0131 geni\u015f spektrumlu etkinlik g\u00f6stermi\u015ftir. Bile\u015fi\u011fin farmakokinetik profili, g\u00fc\u00e7l\u00fc beyin penetrasyonunu vurgulamakta ve onu onkolojide d\u00f6n\u00fc\u015ft\u00fcr\u00fcc\u00fc bir terap\u00f6tik aday olarak konumland\u0131rmaktad\u0131r.<\/span><\/p>\n<\/div><div class=\"fusion-separator fusion-full-width-sep\" style=\"align-self: center;margin-left: auto;margin-right: auto;margin-top:32px;width:100%;\"><div class=\"fusion-separator-border sep-shadow\" style=\"--awb-height:20px;--awb-amount:20px;background:radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-webkit-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-moz-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-o-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);\"><\/div><\/div><div class=\"fusion-image-element\" style=\"text-align:center;--awb-max-width:600px;--awb-caption-title-font-family:var(--h2_typography-font-family);--awb-caption-title-font-weight:var(--h2_typography-font-weight);--awb-caption-title-font-style:var(--h2_typography-font-style);--awb-caption-title-size:var(--h2_typography-font-size);--awb-caption-title-transform:var(--h2_typography-text-transform);--awb-caption-title-line-height:var(--h2_typography-line-height);--awb-caption-title-letter-spacing:var(--h2_typography-letter-spacing);\"><span class=\" fusion-imageframe imageframe-none imageframe-2 hover-type-magnify has-image-magnify fusion-animated\" style=\"border-radius:10px;\" data-animationType=\"fadeInDown\" data-animationDuration=\"0.4\" data-animationOffset=\"top-into-view\" data-magnify-duration=\"400\"><img decoding=\"async\" width=\"1024\" height=\"576\" title=\"only_protein4\" src=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-1024x576.png\" alt class=\"img-responsive wp-image-8998\" srcset=\"https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-200x112.png 200w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-400x225.png 400w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-600x337.png 600w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-800x450.png 800w, https:\/\/www.ortaakarsu.net\/wp-content\/uploads\/only_protein4-1200x675.png 1200w\" sizes=\"(max-width: 640px) 100vw, 1200px\" \/><\/span><\/div><div class=\"fusion-separator fusion-full-width-sep\" style=\"align-self: center;margin-left: auto;margin-right: auto;margin-top:32px;width:100%;\"><div class=\"fusion-separator-border sep-shadow\" style=\"--awb-height:20px;--awb-amount:20px;background:radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-webkit-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-moz-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);background:-o-radial-gradient(ellipse at 50% -50% , var(--awb-color3) 0px, rgba(255, 255, 255, 0) 80%) repeat scroll 0 0 rgba(0, 0, 0, 0);\"><\/div><\/div><div class=\"fusion-title title fusion-title-5 fusion-sep-none fusion-title-text fusion-title-size-four\" style=\"--awb-margin-top-small:10px;--awb-margin-right-small:0px;--awb-margin-bottom-small:10px;--awb-margin-left-small:0px;\"><h4 class=\"fusion-title-heading title-heading-left\" style=\"margin:0;\">G\u00f6rselle\u015ftirmenin Analiz Kolayl\u0131\u011f\u0131 Sa\u011flamas\u0131<\/h4><\/div><div class=\"fusion-text fusion-text-6 awb-text-cols fusion-text-columns-2\" style=\"--awb-columns:2;--awb-column-spacing:2em;--awb-column-min-width:100px;\"><p>Bu video, NST-628&#8217;in BRAF\/MEK kompleksi ile etkile\u015fiminin dinamiklerini g\u00f6rsel olarak yakalayarak hem bilimsel ara\u015ft\u0131rmac\u0131lara hem de bilin\u00e7li izleyicilere mekanizmas\u0131n\u0131n atomik \u00f6l\u00e7ekte anla\u015f\u0131lmas\u0131n\u0131 sa\u011flar. Sim\u00fclasyon, molek\u00fcler yerle\u015ftirme, geli\u015fmi\u015f g\u00f6rselle\u015ftirme teknikleri ve titiz molek\u00fcler dinamik sim\u00fclasyonlar dahil olmak \u00fczere kullan\u0131lan geli\u015fmi\u015f hesaplama y\u00f6ntemlerini vurgulayarak ayr\u0131nt\u0131l\u0131 molek\u00fcler etkile\u015fimleri ortaya koymaktad\u0131r.<\/p>\n<p>NST-628&#8217;in RAF-MEK yola\u011f\u0131n\u0131n kal\u0131c\u0131 inhibisyonunu benzersiz bir \u015fekilde nas\u0131l sa\u011flad\u0131\u011f\u0131n\u0131 g\u00f6steren bu video, onkoloji ara\u015ft\u0131rmalar\u0131, ila\u00e7 ke\u015ffi, yap\u0131sal biyoloji ve molek\u00fcler farmakoloji ile ilgilenen profesyoneller i\u00e7in bir e\u011fitim kayna\u011f\u0131 g\u00f6revi g\u00f6rmektedir. Ayr\u0131ca, \u00e7\u0131\u011f\u0131r a\u00e7an kanser tedavileriyle ilgilenen bilimsel okuryazar bireylere de hitap etmektedir.<\/p>\n<p>Kendine \u00f6zg\u00fc mekanizmas\u0131 ve klinik potansiyeli g\u00f6z \u00f6n\u00fcne al\u0131nd\u0131\u011f\u0131nda, NST-628, RAS ve RAF odakl\u0131 kanserler i\u00e7in terap\u00f6tik stratejileri yeniden tan\u0131mlayabilir ve kar\u015f\u0131lanmam\u0131\u015f kritik t\u0131bbi ihtiya\u00e7lar\u0131 kar\u015f\u0131layabilir. Yenilik\u00e7i kanser tedavileri hakk\u0131nda daha fazla son teknoloji bilimsel g\u00f6rselle\u015ftirme ve g\u00fcncellemeler i\u00e7in bizi izlemeye devam edin ve abone olun.<\/p>\n<\/div><\/div><\/div><div class=\"fusion-layout-column fusion_builder_column fusion-builder-column-5 fusion_builder_column_1_1 1_1 fusion-flex-column fusion-animated\" style=\"--awb-bg-blend:overlay;--awb-bg-size:cover;--awb-width-large:100%;--awb-margin-top-large:0px;--awb-spacing-right-large:0px;--awb-margin-bottom-large:40px;--awb-spacing-left-large:0px;--awb-width-medium:100%;--awb-spacing-right-medium:0px;--awb-spacing-left-medium:0px;--awb-width-small:100%;--awb-spacing-right-small:0px;--awb-spacing-left-small:0px;\" data-animationType=\"fadeInDown\" data-animationDuration=\"0.6\" data-animationOffset=\"top-into-view\"><div class=\"fusion-column-wrapper fusion-column-has-shadow fusion-flex-justify-content-flex-start fusion-content-layout-column\"><div class=\"fusion-sharing-box fusion-sharing-box-1 has-taglines layout-floated layout-medium-floated layout-small-floated\" style=\"background-color:var(--awb-color2);--awb-layout:row;--awb-alignment-small:space-between;\" data-title=\"Aktif B\u00f6lgeye G\u00f6m\u00fcl\u00fc Bir Ligand\u0131n Zamana Ba\u011fl\u0131 Hareketi\" data-description=\"Edible Easter Slime  Recommended for you    MMolek\u00fcler dinamik (MD) sim\u00fclasyonlar\u0131, geleneksel deneysel y\u00f6ntemlere gizli kalan atomik d\u00fczeydeki olaylar\u0131 g\u00f6rselle\u015ftirme ve anlama kapasitemizde devrim yaratm\u0131\u015ft\u0131r. 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