{"id":7571,"date":"2021-08-02T15:41:22","date_gmt":"2021-08-02T12:41:22","guid":{"rendered":"https:\/\/www.ortaakarsu.net\/?p=7571"},"modified":"2025-04-12T16:53:02","modified_gmt":"2025-04-12T13:53:02","slug":"yasmin-dogum-kontrol-hapi-ve-yan-etkileri","status":"publish","type":"post","link":"https:\/\/www.ortaakarsu.net\/?p=7571","title":{"rendered":"Yasmin Do\u011fum Kontrol Hap\u0131 ve Yan Etkileri"},"content":{"rendered":"\r\n<p class=\"wp-block-paragraph\">Drospirenon etken maddesine sahip ila\u00e7, <strong>yasmin do\u011fum kontrol hap\u0131<\/strong> ad\u0131 alt\u0131nda ticari olarak sat\u0131lmaktd\u0131r. Progesteron ve \u00f6strojen i\u00e7eri\u011fine sahip, oral kullan\u0131ma uygun do\u011fum kontrol haplar\u0131na <strong>kombine oral kontraseptif<\/strong> denilmektedir. Yasmin do\u011fum kontrol hap\u0131 bu ila\u00e7 s\u0131n\u0131f\u0131nda yer alan ila\u00e7lardan biridir.<\/p>\r\n\r\n\r\n\r\n<p class=\"wp-block-paragraph\">Yasmin Do\u011fum Kontrol hap\u0131 do\u011fum kontrol\u00fc amac\u0131yla kullan\u0131ld\u0131\u011f\u0131 gibi hormonlara ba\u011fl\u0131 su tutmas\u0131, sivilce, ciltte ya\u011flanma gibi \u015fikayetlerin giderilmesi amac\u0131yla da s\u0131kl\u0131kla kullan\u0131lmaktad\u0131r. Her iki durumda da ilac\u0131n d\u00fczenli ve planl\u0131 kullan\u0131m\u0131 ilac\u0131n etkisini g\u00f6stermesi i\u00e7in gerekli olan birincil \u015fartt\u0131r.<\/p>\r\n\r\n\r\n\r\n<p class=\"wp-block-paragraph\">\u0130lac\u0131n etken maddesi drospirenon steroid yap\u0131s\u0131d\u0131r ve bu bir progestin ilac\u0131d\u0131r. Daha \u00f6nce s\u00f6yledi\u011fimiz gibi hamileli\u011fi \u00f6nlemede kullan\u0131l\u0131r. Ayr\u0131ca menopoz d\u00f6neminde de kullan\u0131m\u0131 mevcuttur. Bu etken maddeye sahip ba\u015fka bir ila\u00e7 olan Yazz do\u011fum kontrol ilac\u0131 hakk\u0131nda daha fazla bilgiye <a href=\"https:\/\/www.ortaakarsu.net\/?p=8025\">Yazz Do\u011fum Kontrol Hap\u0131<\/a> yaz\u0131s\u0131n\u0131 okuyarak sahip olabilirsiniz.<\/p>\r\n\r\n\r\n\r\n\r\n\r\n<h2 class=\"wp-block-heading\">Yasmin Do\u011fum Kontrol Hap\u0131 Kullanan Yorumlar\u0131<\/h2>\r\n\r\n\r\n\r\n<p class=\"wp-block-paragraph\">Klinik \u00e7al\u0131\u015fmalar ve di\u011fer bilimsel ara\u015ft\u0131rmalar ilac\u0131n d\u00fczenli kullan\u0131m\u0131nda hamileli\u011fi engelledi\u011fini ve belirli hastal\u0131klar \u00fczerinde tedavi edici etkileri oldu\u011funu g\u00f6stermektedir. <strong>\u0130lac\u0131 kullananlar\u0131n g\u00f6r\u00fc\u015fleri etkili oldu y\u00f6n\u00fcndedir. Yan etki olarak adet d\u00f6ng\u00fcs\u00fcnde de\u011fi\u015fimlere neden oldu\u011fu s\u0131kl\u0131kla duyulmaktad\u0131r. \u00c7e\u015fitli hormonal de\u011fi\u015fimlerin s\u00f6z konusu olabilece\u011fi s\u0131kl\u0131kla s\u00f6ylenen kullanan yorumlar\u0131ndand\u0131r<\/strong>. T\u00fcm bu veriler b\u00fct\u00fcn olarak de\u011ferlendirildi\u011finde <strong>Yasmin Do\u011fum Kontrol Hap\u0131<\/strong>&#8216;n\u0131n g\u00fcvenle kullan\u0131labilece\u011fi sonucu ortaya \u00e7\u0131kmaktad\u0131r.<\/p>\r\n<p>Ayr\u0131ca ilac\u0131n kullan\u0131m\u0131 i\u00e7in adet d\u00f6ng\u00fclerinin d\u00fczenlenmesi durumu da vard\u0131r. Bu konuda da kullan\u0131c\u0131 yorumlar\u0131 adet d\u00f6ng\u00fclerinin d\u00fczenlendi\u011fi ve rahat bir d\u00f6nem ge\u00e7irdikleri y\u00f6n\u00fcndedir. Yasmin do\u011fum kontrol ilac\u0131n\u0131n \u00f6strojen bazl\u0131 olmas\u0131 bu kullan\u0131m amac\u0131ndaki etkisini ve olumlu kullan\u0131c\u0131 yorumlar\u0131n\u0131 a\u00e7\u0131klamaktad\u0131r.<\/p>\r\n<h3><strong>Olumlu Yorumlar<\/strong><\/h3>\r\n<ul>\r\n<li><strong data-start=\"546\" data-end=\"575\">Adet Sanc\u0131lar\u0131nda Azalma:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kullan\u0131c\u0131lar, Yasmin&#8217;in adet sanc\u0131lar\u0131n\u0131 hafifletti\u011fini ve daha rahat bir d\u00f6nem ge\u00e7irdiklerini belirtmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"392\" data-end=\"422\">Adet D\u00fczeninin Sa\u011flanmas\u0131:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Adet d\u00fczensizli\u011fi ya\u015fayan baz\u0131 kad\u0131nlar, Yasmin kullan\u0131m\u0131yla birlikte adetlerinin d\u00fczenli hale geldi\u011fini ifade etmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"235\" data-end=\"268\">Cilt Problemlerinde \u0130yile\u015fme:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kullan\u0131c\u0131lar, Yasmin&#8217;in sivilce ve cilt ya\u011flanmas\u0131n\u0131 azaltt\u0131\u011f\u0131n\u0131 belirtmi\u015ftir.<\/span><\/li>\r\n<\/ul>\r\n<h3><strong>Olumsuz Yorumlar<\/strong><\/h3>\r\n<ul>\r\n<li><strong data-start=\"722\" data-end=\"756\">Mide Bulant\u0131s\u0131 ve Ba\u015f D\u00f6nmesi:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kullan\u0131c\u0131lar, ilac\u0131n kullan\u0131m\u0131n\u0131n ilk haftalar\u0131nda mide bulant\u0131s\u0131 ve ba\u015f d\u00f6nmesi ya\u015fad\u0131klar\u0131n\u0131 bildirmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"884\" data-end=\"911\">Duygusal Dalgalanmalar:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kad\u0131nlar, Yasmin kullan\u0131m\u0131 s\u0131ras\u0131nda duygusal dalgalanmalar, sinirlilik ve depresif hisler ya\u015fad\u0131klar\u0131n\u0131 ifade etmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"1041\" data-end=\"1067\">Cinsel \u0130stekte Azalma:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kullan\u0131c\u0131lar, ilac\u0131n cinsel istekte azalmaya neden oldu\u011funu belirtmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"1197\" data-end=\"1221\">Kilo De\u011fi\u015fiklikleri:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kad\u0131nlar, Yasmin kullan\u0131m\u0131 s\u0131ras\u0131nda i\u015ftah art\u0131\u015f\u0131 ve kilo al\u0131m\u0131 ya\u015fad\u0131klar\u0131n\u0131 ifade etmi\u015ftir.<\/span><\/li>\r\n<li><strong data-start=\"1351\" data-end=\"1395\">Sa\u00e7 D\u00f6k\u00fclmesi ve V\u00fccut T\u00fcylerinde Art\u0131\u015f:<\/strong> <span class=\"relative -mx-px my-[-0.2rem] rounded-sm px-px py-[0.2rem]\">Baz\u0131 kullan\u0131c\u0131lar, sa\u00e7 d\u00f6k\u00fclmesi ve v\u00fccut t\u00fcylerinde art\u0131\u015f gibi yan etkiler bildirmi\u015ftir.<\/span><\/li>\r\n<\/ul>\r\n<p>\r\n\r\n<\/p>\r\n<h2 class=\"wp-block-heading\">Yasmin Do\u011fum Kontrol Hap\u0131 Yan Etkileri<\/h2>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Yan etkilerinden baz\u0131lar\u0131 \u015fu \u015fekilde s\u0131ralanabilir:<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<ul class=\"wp-block-list\">\r\n<li>Akne(hormon durumundaki ani de\u011fi\u015fikliklere v\u00fccudun verdi\u011fi bir tepki olarak)<\/li>\r\n\r\n\r\n\r\n<li>Ba\u015f a\u011fr\u0131s\u0131(kan dola\u015f\u0131m\u0131ndaki ila\u00e7 y\u00fck\u00fcn\u00fcn lipit a\u011f\u0131rl\u0131kl\u0131 olmas\u0131ndan kaynaklanabildi\u011fi d\u00fc\u015f\u00fcn\u00fclmektedir)<\/li>\r\n\r\n\r\n\r\n<li>Meme Hassasiyeti(\u00f6strojen art\u0131\u015f\u0131 s\u00fct bezlerinde b\u00fcy\u00fcmeyi ve hassasiyeti beraberinde getirir)<\/li>\r\n\r\n\r\n\r\n<li>Kiloda art\u0131\u015f(resept\u00f6r uyar\u0131lmas\u0131 beraberinde i\u015ftah de\u011fi\u015fimlerini beraberinde getirir)<\/li>\r\n\r\n\r\n\r\n<li>Adet d\u00f6ng\u00fcs\u00fcnde zamanlama de\u011fi\u015fiklikleri(yumurta geli\u015fimi \u00f6strojen hormonundaki de\u011fi\u015fimlerden y\u00fcksek oranda etkilenir)<\/li>\r\n<\/ul>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Nadir g\u00f6r\u00fclen yan etkiler ise y\u00fcksek potasyum seviyeleri ve kan p\u0131ht\u0131la\u015fmas\u0131 vard\u0131r. \u00d6zellikle kan p\u0131ht\u0131la\u015fmas\u0131 bu etken maddeyi i\u00e7eren b\u00fct\u00fcn ila\u00e7lar\u0131n prospekt\u00fcs\u00fcnde \u00f6nemli bir yer tutmaktad\u0131r ve olduk\u00e7a \u00f6nemlidir.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Drospirenon sentetik bir progestojen olarak kar\u015f\u0131m\u0131za \u00e7\u0131kmaktad\u0131r. Yani progesteronda oldu\u011fu gibi progesteron resept\u00f6r\u00fcne ba\u011flanmaktad\u0131r. <strong>Drospirenon bir progesteron agonistidir<\/strong>. Drospirenon di\u011fer steroid yap\u0131daki progestinlerden daha fazla biyo uyumlu, progesterona daha fazla benzeyen bir molek\u00fcld\u00fcr.\u00a0<\/p>\r\n<p>\r\n\r\n\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Drospirenone&#8217;in 1976 y\u0131l\u0131nda ilk patent ba\u015fvurusu yap\u0131lm\u0131\u015f ve 2000 y\u0131l\u0131nda t\u0131bbi kullan\u0131ma ge\u00e7mi\u015ftir. Pek \u00e7ok marka ad\u0131 alt\u0131nda do\u011fum kontrol ilac\u0131 olarak s\u0131kl\u0131kla kullan\u0131lmaktad\u0131r. Amerika&#8217;da en \u00e7ok re\u00e7ete edilen ilk iki y\u00fcz ila\u00e7 aras\u0131nda yerini alm\u0131\u015ft\u0131r.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Bu ila\u00e7 farkl\u0131 form\u00fclasyonlar ile kullan\u0131m amac\u0131na g\u00f6re ticari olarak sunulmaktad\u0131r. Baz\u0131 form\u00fclasyonlar \u00f6strodiol gibi hormonlar\u0131 i\u00e7ermektedir. Yasmin do\u011fum kontrol hap\u0131 etinilestradiol ile form\u00fclasyon halinde bulunmaktad\u0131r.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Yeni yaz\u0131lar\u0131m\u0131z\u0131 incelemek i\u00e7in <a href=\"https:\/\/www.ortaakarsu.net\/?p=7959\">Levopront \u2013 Levodropropizin \u2013 \u00d6ks\u00fcr\u00fck \u015eurubu<\/a>, <a href=\"https:\/\/www.ortaakarsu.net\/?p=7861\">Rivoclon Nedir?<\/a>, <a href=\"https:\/\/www.ortaakarsu.net\/?p=7768\">Olanzapin Yan Etkileri ve Kullan\u0131c\u0131 Yorumlar\u0131<\/a> ve <a href=\"https:\/\/www.ortaakarsu.net\/?p=7942\">Amoksisilin Beta Laktamaz \u0130nhibit\u00f6rleri<\/a> yaz\u0131lar\u0131n\u0131 okuyabilirsiniz.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<h2 class=\"wp-block-heading\">Literat\u00fcrdeki \u00c7al\u0131\u015fmalar<\/h2>\r\n<p>\r\n\r\n<\/p>\r\n<figure class=\"wp-block-embed is-type-video is-provider-youtube wp-block-embed-youtube wp-embed-aspect-16-9 wp-has-aspect-ratio\"><\/figure>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Literat\u00fcrde <strong>Yasmin Do\u011fum Kontrol Hap\u0131<\/strong> ile ilgili pek \u00e7ok klinik ve deneysel \u00e7al\u0131\u015fma mevcuttur. Bu \u00e7al\u0131\u015fmalardan baz\u0131lar\u0131n\u0131n \u00f6zet k\u0131s\u0131mlar\u0131n\u0131 derledik ve bir yaz\u0131 haline getirdik. E\u011fer bir ara\u015ft\u0131rmac\u0131ysan\u0131z kaynak linklerinden as\u0131l yaz\u0131ya ve yaz\u0131n\u0131n tamam\u0131na ula\u015fabilirsiniz.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<h3 class=\"wp-block-heading\">Yasmin Do\u011fum Kontrol Hap\u0131n\u0131n Etkileri<\/h3>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Di\u011fer progestojenlerden farkl\u0131 olarak, bir spironolakton analo\u011fu olan drospirenon, \u00f6zellikle antimineralokortikoid ve antiandrojenik aktiviteler a\u00e7\u0131s\u0131ndan endojen progesterona benzer biyokimyasal ve farmakolojik profillere sahiptir. Drospirenon, renin-anjiyotensin-aldosteron sisteminin \u00f6strojen kaynakl\u0131 stim\u00fclasyonuna kar\u015f\u0131 koyar ve testosteronun androjen resept\u00f6rlerine ba\u011flanmas\u0131n\u0131 engeller. Bu \u00f6zelliklerinden dolay\u0131 v\u00fccut a\u011f\u0131rl\u0131\u011f\u0131n\u0131, kan bas\u0131nc\u0131n\u0131 ve d\u00fc\u015f\u00fck yo\u011funluklu lipoprotein d\u00fczeylerini d\u00fc\u015f\u00fcrme ve y\u00fcksek yo\u011funluklu lipoprotein d\u00fczeylerini art\u0131rma potansiyeline sahiptir. Bir kombinasyon oral kontraseptif olarak, etinil estradiol ile drospirenon etkilidir ve a\u011f\u0131rl\u0131k ve lipid seviyeleri \u00fczerinde olumlu etkileri vard\u0131r. Ek olarak, di\u011fer kombine oral kontraseptiflerle yayg\u0131n olarak g\u00f6zlenen menstr\u00fcel ili\u015fkili semptomlar\u0131 (\u00f6rn. olumsuz duygulan\u0131m ve su tutulmas\u0131) hafifletir. Biyokimyasal ve farmakodinamik verilere dayanarak, drospirenon \u015fu anda mevcut olan progestojenlere uygun bir alternatif gibi g\u00f6r\u00fcnmektedir. Kaynak:<a href=\"https:\/\/doi.org\/10.1016\/S0010-7824(00)00133-5\" target=\"_blank\" rel=\"noreferrer noopener\">https:\/\/doi.org\/10.1016\/S0010-7824(00)00133-5<\/a><\/p>\r\n<h3 class=\"\" data-start=\"710\" data-end=\"798\"><strong data-start=\"717\" data-end=\"798\">Anti-Androjenik Etkisi ile Polikistik Over Sendromu (PCOS) \u00dczerindeki Rol\u00fc<\/strong><\/h3>\r\n<ul data-start=\"799\" data-end=\"973\">\r\n<li class=\"\" data-start=\"799\" data-end=\"871\">\r\n<p class=\"\" data-start=\"801\" data-end=\"871\">PCOS hastalar\u0131 i\u00e7in \u00f6nerilen do\u011fum kontrol ila\u00e7lar\u0131 aras\u0131nda yer al\u0131r.<\/p>\r\n<\/li>\r\n<li class=\"\" data-start=\"872\" data-end=\"973\">\r\n<p class=\"\" data-start=\"874\" data-end=\"973\">Testosteron etkilerini bask\u0131layarak t\u00fcylenme (hirsutizm) ve akne gibi \u015fikayetlerde iyile\u015fme sa\u011flar.<\/p>\r\n<\/li>\r\n<\/ul>\r\n<h3 class=\"\" data-start=\"1377\" data-end=\"1433\"><strong data-start=\"1384\" data-end=\"1433\">Yasmin ve Ven\u00f6z Tromboembolizm (VTE) Riski<\/strong><\/h3>\r\n<ul data-start=\"1434\" data-end=\"1795\">\r\n<li class=\"\" data-start=\"1434\" data-end=\"1540\">\r\n<p class=\"\" data-start=\"1436\" data-end=\"1540\">Yasmin, di\u011fer do\u011fum kontrol haplar\u0131na g\u00f6re daha d\u00fc\u015f\u00fck ancak <strong data-start=\"1496\" data-end=\"1533\">hala anlaml\u0131 bir p\u0131ht\u0131la\u015fma riski<\/strong> ta\u015f\u0131r.<\/p>\r\n<\/li>\r\n<li class=\"\" data-start=\"1541\" data-end=\"1636\">\r\n<p class=\"\" data-start=\"1543\" data-end=\"1636\">Bu nedenle sigara i\u00e7en, 35 ya\u015f \u00fcst\u00fc veya p\u0131ht\u0131 \u00f6yk\u00fcs\u00fc olan bireyler i\u00e7in <strong data-start=\"1616\" data-end=\"1626\">riskli<\/strong> olabilir.<\/p>\r\n<\/li>\r\n<\/ul>\r\n<h3 class=\"\" data-start=\"1802\" data-end=\"1862\"><strong data-start=\"1809\" data-end=\"1862\">Kullan\u0131m Kolayl\u0131\u011f\u0131 ve Kullan\u0131c\u0131 Uyumuna Etkisi<\/strong><\/h3>\r\n<ul data-start=\"1863\" data-end=\"2087\">\r\n<li class=\"\" data-start=\"1863\" data-end=\"1980\">\r\n<p class=\"\" data-start=\"1865\" data-end=\"1980\">21+7 g\u00fcn kullan\u0131m \u015femas\u0131 ile adet d\u00fczenini taklit eder. Bu, <strong data-start=\"1925\" data-end=\"1972\">duygusal olarak g\u00fcven verici bir d\u00fczenlilik<\/strong> sa\u011flar.<\/p>\r\n<\/li>\r\n<li class=\"\" data-start=\"1981\" data-end=\"2087\">\r\n<p class=\"\" data-start=\"1983\" data-end=\"2087\">Re\u00e7eteli sat\u0131lmas\u0131 ve doktor kontrol\u00fc gerektirmesi, kullan\u0131c\u0131lar\u0131n ilac\u0131 bilin\u00e7li kullanmalar\u0131n\u0131 sa\u011flar.<\/p>\r\n<\/li>\r\n<\/ul>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">\r\n\r\n<\/p>\r\n<h3 class=\"wp-block-heading\">Di\u011fer Do\u011fum Kontrol Haplar\u0131, Tedavide Kullan\u0131mlar\u0131 ve Yasmin Do\u011fum Kontrol Yap\u0131<\/h3>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Do\u011fum kontrol\u00fc ve hormon replasman tedavisinde (HRT) kullan\u0131lan progestinlerin farmakolojik \u00f6zellikleri, t\u00fcretildikleri molek\u00fcllere ba\u011fl\u0131 olarak de\u011fi\u015fir. \u00c7ok k\u00fc\u00e7\u00fck yap\u0131sal de\u011fi\u015fiklikler, etkilerde \u00f6nemli farkl\u0131l\u0131klara neden olabilir. Halihaz\u0131rda mevcut olan progestinlerin, progesteron resept\u00f6rlerine, PR-A veya PR-B&#8217;ye spesifik olarak ba\u011flan\u0131p ba\u011flanamad\u0131\u011f\u0131 belirsizdir. Progesteron resept\u00f6r\u00fcn\u00fcn bir veya di\u011fer izoformlar\u0131na daha spesifik ba\u011flanman\u0131n klinik \u00f6nemi hala bilinmemektedir. \u0130yile\u015ftirilmi\u015f resept\u00f6r se\u00e7icilik profilleri ile yeni nesil progestinlerin geli\u015ftirilmesi b\u00fcy\u00fck bir zorluk olmu\u015ftur. Steroidal ve steroidal olmayan progesteron agonistleri de sentezlenmi\u015ftir, ancak bu molek\u00fcller geli\u015fimin \u00e7ok erken bir a\u015famas\u0131ndad\u0131r. Son on y\u0131lda dienogest, drospirenon, Nestorone, nomegestrol asetat ve trimegeston dahil olmak \u00fczere birka\u00e7 yeni progestin sentezlendi. Drospirenon, spirolaktondan t\u00fcretilmesiyle klasik progestinlerden farkl\u0131d\u0131r. Drospirenonun ana etkisi, antimineralocorticoid aktivitesidir. Bu \u00f6zelli\u011fi sayesinde, drospirenon, tuz ve su tutulmas\u0131n\u0131n azalmas\u0131na ve dolay\u0131s\u0131yla kan bas\u0131nc\u0131n\u0131n d\u00fc\u015fmesine neden olur. Drospirenonun mineralokortikoid resept\u00f6r\u00fcne afinitesi, do\u011fal olarak olu\u015fan mineralokortikoid olan aldosteronun yakla\u015f\u0131k be\u015f kat\u0131d\u0131r.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">Ek olarak, drospirenonun androjenik etkisi yoktur, ancak k\u0131smi antiandrojenik aktivite sergiler; antiandrojenik g\u00fcc\u00fc, en g\u00fc\u00e7l\u00fc antiandrojenik aktiviteye sahip progestin olan siproteron asetat\u0131n yakla\u015f\u0131k %30&#8217;udur. Birka\u00e7 yeni progestin taraf\u0131ndan payla\u015f\u0131lan bu \u00f6zellik, androjenlerin postmenopozal kad\u0131nlarda sa\u00e7 b\u00fcy\u00fcmesi, lipid de\u011fi\u015fiklikleri, ins\u00fclin ve muhtemelen v\u00fccut kompozisyonu \u00fczerindeki olumsuz etkisini ortadan kald\u0131rabilir. Drospirenon uzun bir terminal yar\u0131 \u00f6mre (yakla\u015f\u0131k 32 saat) sahiptir ve biyoyararlan\u0131m\u0131 yakla\u015f\u0131k %76&#8217;d\u0131r. Progesteronunkine \u00e7ok benzer farmakodinamik \u00f6zelliklere sahip olan Drospirenon, kombine bir oral kontraseptif olarak geli\u015ftirilmi\u015ftir (30 \u03bcg etinilestradiol\/3 mg drospirenon; Yasmin\u00ae, Schering AG, Berlin, Almanya). Drospirenon, bir HRT preparat\u0131 olarak estradiol ile kombinasyon halinde de mevcuttur (1 mg 17\u03b2-estradiol\/2 mg drospirenon; Angeliq\u00ae, Schering AG). Kaynak: <a href=\"https:\/\/doi.org\/10.1080\/13697130500330382\">https:\/\/doi.org\/10.1080\/13697130500330382<\/a><\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p class=\"wp-block-paragraph\">L\u00fctfen kulland\u0131\u011f\u0131n\u0131z ila\u00e7lar\u0131 doktorunuzun bilgisi d\u0131\u015f\u0131nda kombine etmeyiniz ve \u00f6nerilen dozu a\u015fmay\u0131n\u0131z. \u0130la\u00e7lar\u0131n\u0131z\u0131 her zaman doktorunuzun re\u00e7ete etti\u011fi \u015fekilde kullan\u0131n\u0131z. Buna <strong>yasmin do\u011fum kontrol hap\u0131<\/strong> da dahil.<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p>\r\n\r\n<\/p>\r\n<p><\/p>","protected":false},"excerpt":{"rendered":"<p>Drospirenon etken maddesine sahip ila\u00e7, yasmin do\u011fum kontrol hap\u0131 ad\u0131  [&#8230;]<\/p>\n","protected":false},"author":1,"featured_media":9351,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_acf_changed":false,"footnotes":""},"categories":[122],"tags":[110,254,256,255,125,143,9,153,202,251,219,253,336],"class_list":["post-7571","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-molekul","tag-biyokimya","tag-dogum-kontrol-hapi","tag-dogum-kontrolu","tag-drospirenon","tag-ilac","tag-ilac-gelistirme","tag-ilac-tasarimi","tag-ostrojen","tag-reseptor","tag-steroid","tag-yan-etki","tag-yasmin-dogum-kontrol-hapi","tag-yazz-dogum-kontrol-hapi"],"acf":[],"_links":{"self":[{"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/posts\/7571","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=7571"}],"version-history":[{"count":23,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/posts\/7571\/revisions"}],"predecessor-version":[{"id":9287,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/posts\/7571\/revisions\/9287"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=\/wp\/v2\/media\/9351"}],"wp:attachment":[{"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=7571"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=%2Fwp%2Fv2%2Fcategories&post=7571"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/www.ortaakarsu.net\/index.php?rest_route=%2Fwp%2Fv2%2Ftags&post=7571"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}